Drugs that should not be co-administered with ritonavir/Norvirtm

(from the "Contraindications" section of the ritonavir/Norvirtm drug insert)

Contraindicated due to risks of arrhythmias ("irregularity or loss of rhythm, particularly the heartbeat"), hematologic ("blood") abnormalities, seizures or other potentially serious adverse affects:

  1. amiodarone (Cordaronetm)
  2. astemizole (Hismanaltm)
  3. bepridil (Vascortm)
  4. bupropion (Wellbutrintm)
  5. cisapride (Propulsidtm)
  6. clozapine (Clozariltm)
  7. encainide (Enkaidtm)
  8. flecainide (Tambocortm)
  9. meperidine (Demeroltm, Mepergantm, Meperidinetm)
  10. piroxicam (Feldenetm)
  11. propafenone (Rythmoltm)
  12. propoxyphene (Darvontm, Propoxyphenetm, Wygesictm)
  13. quinidine (Duraquintm, Quinaglutetm, Quinalantm, Quinidinetm)
  14. rifabutin (Mycobutintm) - for Mycobacterium avium complex (MAC) prophylaxis
  15. terfenadine (Seldanetm)

Contraindicated due to potential for extreme sedation and respiratory depression:

  1. alprazolam (Xanaxtm)
  2. clorazepate (Clorazepatetm, Gen-XENEtm, Tranxenetm)
  3. diazepam (Diazepamtm, Valiumtm, Valreleasetm)
  4. estazolam (ProSomtm)
  5. flurazepam (Dalmanetm, Flurazepamtm)
  6. midazolam (Versedtm)
  7. triazolam (Halciontm)
  8. zolpidem (Ambientm)

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